SCHEMBL8538552

SCHEMBL8538552

O=C1NCCN(c2ccc(OC(F)(F)C(F)F)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
LIPE Q05469 9/20 0.37
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
MMP13 P45452 1/20 0.34
MMP14 P50281 1/20 0.34
KCNH2 Q12809 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ABL1 P00519 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
DPP4 P27487 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8584198 0.87 LIPE (0.39) SCN5ASCN9ALIPEPIM1PIM2
SCHEMBL8536210 0.82 HTT (0.40) LIPEMMP13MMP14ALDH1A1
SCHEMBL10497873 0.75 SCN5A (0.46) SCN5ASCN9AABL1HCRTR1HCRTR2
SCHEMBL20956958 0.74 LIPE (0.49) LIPEPOLBL3MBTL1
SCHEMBL8540845 0.73 ALDH1A1 (0.44) SCN5ASCN9ALIPEPIM1PIM2
SCHEMBL8584196 0.72 SCN5A (0.39) SCN5ASCN9ALIPEMMP13MMP14
SCHEMBL8674715 0.71 LIPE (0.39) SCN9ALIPEMMP13POLBL3MBTL1
SCHEMBL6224361 0.71 NPC1 (0.50) POLBALDH1A1
SCHEMBL3937241 0.71 ADRB1 (0.56) ALDH1A1
SCHEMBL8668327 0.69 CMA1 (0.39) LIPEPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792780-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-11 US disclosed
EP-0657449-B1 Azole compounds, their production and use as antifungal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-04-08 EP disclosed
US-5545652-A Triazole and imidazole compounds and their use as antifungal therapeutic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-13 US disclosed
EP-0657449-A1 Azole compounds, their production and use as antifungal agents Takeda Chemical Industries, Ltd. (JP) 1995-06-14 EP disclosed