SCHEMBL8540865

SCHEMBL8540865

Oc1ccc(C2CNc3ccccc32)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.41
DRD1 P21728 5/20 0.41
DRD2 P14416 4/20 0.41
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
JAK2 O60674 1/20 0.38
KDM4E B2RXH2 3/20 0.38
RECQL P46063 3/20 0.38
BLM P54132 2/20 0.38
GAA P10253 1/20 0.38
AR P10275 1/20 0.38
IDE P14735 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4001774 0.85 MEN1 (0.52) DRD1DRD2KMT2AMEN1CYP3A4
Hydrochloric Acid SCHEMBL11553849 0.83 MEN1 (0.50) DRD1DRD2KMT2AMEN1CYP3A4
SCHEMBL11601875 0.83 SLC6A2 (0.39) ESR2DRD1DRD2KMT2AMEN1
SCHEMBL5871368 0.82 PRCP (0.42) KMT2AMEN1CYP3A4CYP2D6JAK2
SCHEMBL11516181 0.82 SLC6A2 (0.44) SLC6A2SLC6A4HTR2BSLC6A3
SCHEMBL8485182 0.81 DRD2 (0.41) DRD1DRD2KMT2AMEN1GAA
SCHEMBL8537530 0.79 DRD1 (0.56) DRD1DRD2KMT2AMEN1CYP3A4
SCHEMBL8540456 0.78 PAX8 (0.47) KMT2AMEN1JAK2KDM4EGAA
SCHEMBL8493961 0.78 MEN1 (0.42) DRD1KMT2AMEN1CYP3A4CYP2D6
Formamide SCHEMBL11551135 0.76 MEN1 (0.44) KMT2AMEN1CYP3A4CYP2D6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721949-B1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE CO (JP) 1998-01-07 EP disclosed
US-5677326-A GASTROINTESTINAL DISORDERS TOKYO TANABE COMPANY LIMITED (JP) 1997-10-14 US disclosed
EP-0721949-A1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE COMPANY LIMITED (JP) 1996-07-17 EP disclosed