SCHEMBL8540913

SCHEMBL8540913

Oc1ccc(-c2ccc(-c3ncc[nH]3)cc2)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.49
ESR2 Q92731 6/20 0.49
NISCH Q9Y2I1 2/20 0.47
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MTOR P42345 1/20 0.46
ADK P55263 1/20 0.46
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
CDK2 P24941 2/20 0.43
CDK4 P11802 1/20 0.43
CCNA2 P20248 1/20 0.43
CCND1 P24385 1/20 0.43
CCND3 P30281 1/20 0.43
JAK2 O60674 1/20 0.43
JAK1 P23458 1/20 0.43
TYK2 P29597 1/20 0.43
JAK3 P52333 1/20 0.43
CCNE1 P24864 1/20 0.41
SMPD3 Q9NY59 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL183153 0.80 NISCH (0.64) ESR1ESR2NISCHKDM4EALDH1A1
SCHEMBL9730414 0.80 NISCH (0.47) NISCHKDM4EALDH1A1MTORADK
SCHEMBL8537911 0.77 AMY1A (0.45) ESR1NISCHKDM4EALDH1A1MTOR
SCHEMBL3684267 0.76 ESR1 (0.70) ESR1ESR2HSD17B1HSD17B2
SCHEMBL8541165 0.75 NISCH (0.53) NISCHKDM4EALDH1A1MTORADK
SCHEMBL31429641 0.75 GUSB (0.45) NISCHKDM4EALDH1A1MTORADK
SCHEMBL8540911 0.75 GUSB (0.45) NISCHKDM4EALDH1A1MTORADK
SCHEMBL8535895 0.74 NISCH (0.49) ESR1ESR2NISCHKDM4EALDH1A1
SCHEMBL722191 0.74 NISCH (0.78) NISCHKDM4EALDH1A1MTORADK
SCHEMBL482165 0.73 NISCH (0.64) NISCHKDM4EALDH1A1MTORADK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed