SCHEMBL8540941

SCHEMBL8540941

CC(C)(C)OC(=O)N1CCN(Cc2cccc(C#N)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.59
CHRM4 P08173 2/20 0.51
GLS O94925 2/20 0.49
NSD2 O96028 1/20 0.49
RORC P51449 1/20 0.47
GPR6 P46095 2/20 0.47
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
MGLL Q99685 1/20 0.46
GPR119 Q8TDV5 2/20 0.46
HRH2 P25021 1/20 0.45
HRH1 P35367 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29809169 1.00 FAAH (0.59) FAAHCHRM4GLSNSD2RORC
SCHEMBL1632572 0.93 FAAH (0.53) FAAHCHRM4GLSNSD2RORC
SCHEMBL29121436 0.89 KCNH2 (0.54) FAAHCHRM4NSD2DRD2DRD3
SCHEMBL23334597 0.88 GLS (0.49) FAAHCHRM4GLSNSD2CHRM2
SCHEMBL1066770 0.85 CYP3A4 (0.60) FAAHNSD2GPR119HRH1
SCHEMBL3912590 0.84 FAAH (0.44) FAAHCHRM4MGLLGPR119
SCHEMBL23552038 0.83 VEGFA (0.48) FAAHCHRM4NSD2GPR6GPR119
SCHEMBL2194827 0.83 KDM1A (0.57) CHRM4GLSCHRM2CHRM1CHRM3
SCHEMBL4837787 0.83 GLS (0.54) CHRM4GLSCHRM2CHRM1CHRM3
SCHEMBL8540779 0.83 ALDH1A1 (0.63) FAAHGLSCHRM2CHRM3GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed
WO-2022161420-A1 CLASS OF HETEROAROMATIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊石医药科技有限公司 2022-08-04 WO disclosed
CN-114805341-A Aromatic heterocyclic compounds and preparation method and application thereof 上海翊石医药科技有限公司 2022-07-29 CN disclosed