SCHEMBL8543766

SCHEMBL8543766

CC(=O)NC(=O)c1cccc(N)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HSD17B10 Q99714 1/20 0.53
PBRM1 Q86U86 1/20 0.52
KDM4C Q9H3R0 1/20 0.51
MAPT P10636 2/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
PTGS1 P23219 1/20 0.49
MITF O75030 1/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
MTOR P42345 2/20 0.46
HDAC1 Q13547 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29944867 0.85 HDAC8 (0.63) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL520073 0.85 HDAC8 (0.63) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL7867966 0.84 ALDH1A1 (0.54) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL7188655 0.83 SMN1; SMN2 (0.54) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL6999270 0.83 PBRM1 (0.58) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL9921285 0.80 SMN1; SMN2 (0.59) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL11593734 0.80 PTGS1 (0.67) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL8297913 0.80 ALDH1A1 (0.54) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL294944 0.79 KDM4E (0.66) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10
SCHEMBL6159659 0.79 KDM4E (0.62) ALDH1A1KDM4ESMN1; SMN2NPSR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508796-B1 Cholecystokinin antagonists MERCK & CO INC (US) 1998-07-08 EP disclosed
US-5220018-A Benzodiazepine derivatives MERCK & CO., INC. (US) 1993-06-15 US disclosed
EP-0508796-A1 Cholecystokinin antagonists MERCK & CO. INC. (US) 1992-10-14 EP disclosed