SCHEMBL8544758

SCHEMBL8544758

COC(=O)CCc1[nH]c2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2c1Cc1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
GAA P10253 4/20 0.48
TSHR P16473 1/20 0.48
HTT P42858 1/20 0.48
GFER P55789 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
ITK Q08881 1/20 0.43
KIT P10721 2/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
ERAP1 Q9NZ08 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538927 0.92 MEN1 (0.49) ALDH1A1GAATSHRHTTGFER
SCHEMBL8543376 0.92 AURKA (0.46) ALDH1A1GAATSHRHTTGFER
SCHEMBL8543854 0.91 ALDH1A1 (0.54) ALDH1A1GAATSHRHTTGFER
SCHEMBL8541706 0.91 MEN1 (0.43) ALDH1A1GAATSHRHTTGFER
SCHEMBL8537546 0.85 MEN1 (0.51) ALDH1A1GAAGFERHSD17B10MEN1
SCHEMBL8543931 0.83 BRD4 (0.46) ALDH1A1POLB
SCHEMBL8543318 0.81 MEN1 (0.45) ALDH1A1MEN1KMT2AMAPT
SCHEMBL8539181 0.75 HTR6 (0.56) MEN1KMT2AMAPTKDM4E
SCHEMBL8538700 0.75 TBXAS1 (0.55) ALDH1A1MEN1KMT2A
SCHEMBL8539179 0.74 POLB (0.47) ALDH1A1GAATSHRHTTGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715627-B1 INDOLE DERIVATIVES AS THROMBOXANE A2 ANTAGONISTS PFIZER LTD (GB) 1998-09-09 EP claimed