SCHEMBL8544949

SCHEMBL8544949

Cn1c(=O)oc2cc(C(=O)CCN3CCC(Cc4ccccc4)CC3)ccc21

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.55
GRIN2D O15399 1/20 0.55
GRIN3B O60391 1/20 0.55
GRIN1 Q05586 1/20 0.55
GRIN2A Q12879 1/20 0.55
GRIN2C Q14957 1/20 0.55
GRIN3A Q8TCU5 1/20 0.55
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220636 0.91 ACHE (0.61) ALDH1A1HPGD
SCHEMBL10394036 0.86 ACHE (0.65) ALDH1A1HPGD
SCHEMBL8870163 0.83 SIGMAR1 (0.64) ALDH1A1
SCHEMBL8545288 0.82 GRIN1 (0.62) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL10392907 0.82 ALDH1A1 (0.56) ALDH1A1HPGD
SCHEMBL8546370 0.80 GRIN1 (0.82) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8871026 0.80 SIGMAR1 (0.66) GRIN2B
SCHEMBL9464085 0.80 ALDH1A1 (0.56) ALDH1A1HPGD
SCHEMBL11218131 0.78 MEN1 (0.58) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12123850 0.78 ACHE (0.78) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed