SCHEMBL8549581

SCHEMBL8549581

CN(CCO)C(=O)c1ccc2c(c1)CCOC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 5/20 0.43
HDAC4 P56524 1/20 0.39
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RAB9A P51151 1/20 0.36
AKR1C3 P42330 1/20 0.35
PIR O00625 1/20 0.35
ROCK2 O75116 1/20 0.35
PDK1 Q15118 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
ACACB O00763 1/20 0.34
CNR1 P21554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554148 0.88 EGFR (0.36) PDK2ALDH1A1HPGDGAATSHR
SCHEMBL7092149 0.83 DRD2 (0.40) PDK2ALDH1A1HPGDTSHRMEN1
SCHEMBL8551623 0.82 RAB9A (0.38) PDK2ALDH1A1HPGDGAATSHR
SCHEMBL8550687 0.77 DRD4 (0.48) ALDH1A1TSHRKMT2A
SCHEMBL8549471 0.77 DRD4 (0.48)
SCHEMBL8551575 0.77 DRD4 (0.48) ALDH1A1
SCHEMBL8553551 0.77 DRD4 (0.48)
SCHEMBL8550252 0.76 DRD4 (0.59)
SCHEMBL8549845 0.76 HRH3 (0.49)
SCHEMBL8549100 0.75 DRD4 (0.47) GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed