SCHEMBL8549631

SCHEMBL8549631

NCCc1cn(CCN2CCN(c3ccc(Cl)c(Cl)c3)CC2)c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 6/20 0.49
ADRA1A P35348 5/20 0.49
ADRA1B P35368 4/20 0.49
ALDH1A1 P00352 1/20 0.48
HTT P42858 1/20 0.48
NCOA1 Q15788 1/20 0.48
NCOA3 Q9Y6Q9 1/20 0.48
HTR6 P50406 3/20 0.47
HTR1A P08908 4/20 0.43
HTR2A P28223 3/20 0.43
HTR7 P34969 2/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
ALOX12 P18054 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
DRD2 P14416 5/20 0.42
DRD4 P21917 3/20 0.41
DRD1 P21728 2/20 0.41
DRD3 P35462 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8757616 0.79 HTR2A (0.55) ALDH1A1HTR6HTR2A
SCHEMBL8757614 0.78 HTR2A (0.54) HTR6HTR2A
SCHEMBL9501537 0.78 HTR2A (0.54) HTR2A
SCHEMBL5185937 0.77 MAPT (0.60) ALDH1A1HTTHTR6HTR1AHTR2A
SCHEMBL8618152 0.77 ADRA1D (0.49) ADRA1DADRA1AADRA1BHTR6HTR1A
SCHEMBL8546269 0.77 ADRA1D (0.49) ADRA1DADRA1AADRA1BALDH1A1HTT
SCHEMBL8758865 0.73 ALDH1A1 (0.62) ALDH1A1HTTNCOA1NCOA3HTR6
SCHEMBL5186059 0.72 CYP2D6 (0.59) HTR6HTR1AHTR2AHTR7LMNA
SCHEMBL5185949 0.71 LMNA (0.55) HTR6HTR1AHTR2AHTR7LMNA
SCHEMBL5187801 0.70 KCNH2 (0.56) HTR6HTR1AHTR2AHTR7LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677042-B1 SELECTIVE LIGANDS OF 5HT1D-5HT1B RECEPTORS DERIVED FROM INDOLE-PIPERAZINE USEFUL AS MEDICAMENTS PF MEDICAMENT (FR) 1998-07-22 EP claimed
EP-0677042-B1 SELECTIVE LIGANDS OF 5HT1D-5HT1B RECEPTORS DERIVED FROM INDOLE-PIPERAZINE USEFUL AS MEDICAMENTS PF MEDICAMENT (FR) 1998-07-22 EP disclosed