SCHEMBL8618152

SCHEMBL8618152

NCCc1cn(CCN2CCN(c3cccc4ccccc34)CC2)c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 6/20 0.49
ADRA1A P35348 3/20 0.48
HTR1A P08908 7/20 0.46
HTR2A P28223 3/20 0.46
ADRA1B P35368 2/20 0.46
DRD2 P14416 2/20 0.46
DRD1 P21728 2/20 0.46
HTR2C P28335 2/20 0.46
HTR3A P46098 1/20 0.46
HTR7 P34969 6/20 0.45
CNR1 P21554 1/20 0.45
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546269 0.86 ADRA1D (0.49) ADRA1DADRA1AHTR1AHTR2AADRA1B
SCHEMBL8757616 0.81 HTR2A (0.55) HTR2ACNR1HTR6
SCHEMBL240727 0.81 HTR1A (0.55) ADRA1DADRA1AHTR1AHTR2AADRA1B
SCHEMBL8757614 0.80 HTR2A (0.54) HTR2ACNR1HTR6
SCHEMBL9501537 0.80 HTR2A (0.54) HTR2ACNR1
SCHEMBL8549631 0.77 ADRA1D (0.49) ADRA1DADRA1AHTR1AHTR2AADRA1B
SCHEMBL5187310 0.76 HTR1A (0.60) ADRA1DADRA1AHTR1AHTR2AADRA1B
SCHEMBL5366461 0.75 HTR1A (0.62) HTR1AHTR2ADRD2HTR2CHTR7
SCHEMBL5187168 0.74 HTR1A (0.62) HTR1AHTR2ADRD2HTR2CHTR7
SCHEMBL28374901 0.73 HTR7 (0.56) HTR1AHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677042-B1 SELECTIVE LIGANDS OF 5HT1D-5HT1B RECEPTORS DERIVED FROM INDOLE-PIPERAZINE USEFUL AS MEDICAMENTS PF MEDICAMENT (FR) 1998-07-22 EP claimed
EP-0677042-B1 SELECTIVE LIGANDS OF 5HT1D-5HT1B RECEPTORS DERIVED FROM INDOLE-PIPERAZINE USEFUL AS MEDICAMENTS PF MEDICAMENT (FR) 1998-07-22 EP disclosed