SCHEMBL8549864

SCHEMBL8549864

CS(=O)(=O)OCC1CCN(C(=O)c2ccccc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.56
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51
CA14 Q9ULX7 1/20 0.51
KMT2A Q03164 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
MEN1 O00255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418666 0.88 HDAC3 (0.55) ACHECA12CA1CA2CA7
SCHEMBL9491300 0.84 LMNA (0.54) ACHECA12CA1CA2CA7
SCHEMBL9928308 0.83 ACHE (0.62) ACHEKMT2AHDAC3HDAC4HDAC1
SCHEMBL460173 0.80 SMN1; SMN2 (0.61) KMT2AMEN1SMN1; SMN2
SCHEMBL3533847 0.79 ALDH1A1 (0.35) KMT2AMEN1L3MBTL1
SCHEMBL2780484 0.79 CARM1 (0.61) ACHEKMT2AHDAC3HDAC4HDAC1
SCHEMBL11394317 0.79 KCNA5 (0.58) ACHEHDAC3HDAC4HDAC1HDAC7
SCHEMBL12538923 0.79 ACHE (0.60) ACHECA12CA1CA2CA7
SCHEMBL2618044 0.78 ACHE (0.68) ACHEKMT2AHDAC3HDAC4HDAC1
SCHEMBL5636471 0.77 CHRNB2 (0.49) CA2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed