SCHEMBL8550262

SCHEMBL8550262

O=C(NCc1ccc(Cc2ccc(CNC(=O)NOCc3ccccc3)cc2)cc1)NOCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
EPHX1 P07099 1/20 0.49
CFD P00746 1/20 0.48
PTPN1 P18031 1/20 0.48
TP53 P04637 1/20 0.47
PLAU P00749 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
EPHX2 P34913 1/20 0.46
PPIB P23284 1/20 0.46
PPID Q08752 1/20 0.46
PPIG Q13427 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27537790 0.94 NPC1 (0.59) NPC1RAB9ASMN1; SMN2EPHX1CFD
SCHEMBL8547013 0.88 HPGD (0.57) NPC1RAB9ASMN1; SMN2EPHX1GAA
SCHEMBL8549654 0.84 CARM1 (0.51) NPC1RAB9ASMN1; SMN2PTPN1ALDH1A1
SCHEMBL8546557 0.83 LMNA (0.53) NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL8546499 0.82 HPGD (0.51) SMN1; SMN2KDM4EALDH1A1
SCHEMBL1990363 0.81 NPC1 (0.69) NPC1RAB9AALDH1A1EPHX2
SCHEMBL690027 0.80 NPC1 (0.59) NPC1RAB9AALDH1A1EPHX2CYP1A2
SCHEMBL8549624 0.80 HPGD (0.49) NPC1RAB9ASMN1; SMN2
SCHEMBL8550343 0.80 HSD17B10 (0.46) EPHX1ALDH1A1EPHX2TSHR
SCHEMBL8549404 0.79 HTR2C (0.49) NPC1RAB9AEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed