SCHEMBL8550733

SCHEMBL8550733

O=C(OC1CCN(Cc2ccccc2)CC1)c1ccc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.61
NPSR1 Q6W5P4 1/20 0.61
SIGMAR1 Q99720 5/20 0.48
HPD P32754 1/20 0.47
SERPINE1 P05121 1/20 0.47
FAAH O00519 1/20 0.46
ACHE P22303 1/20 0.46
BCHE P06276 1/20 0.46
UBE2M P61081 1/20 0.46
DCUN1D1 Q96GG9 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8554803 0.99 MAPK1 (0.60) MAPK1NPSR1SIGMAR1HPDSERPINE1
SCHEMBL8550623 0.85 BCHE (0.48) MAPK1SIGMAR1FAAHACHEBCHE
SCHEMBL8553874 0.85 BCHE (0.48) MAPK1NPSR1SIGMAR1FAAHACHE
SCHEMBL8552219 0.85 SIGMAR1 (0.55) MAPK1SIGMAR1BCHE
Hydrochloric Acid SCHEMBL8551753 0.84 BCHE (0.47) MAPK1SIGMAR1FAAHACHEBCHE
Hydrochloric Acid SCHEMBL8551803 0.84 BCHE (0.47) MAPK1NPSR1SIGMAR1FAAHACHE
SCHEMBL8555277 0.84 SIGMAR1 (0.51) SIGMAR1ACHEBCHEUBE2MDCUN1D1
Hydrochloric Acid SCHEMBL8555949 0.84 SIGMAR1 (0.54) MAPK1SIGMAR1BCHE
Hydrochloric Acid SCHEMBL8681759 0.83 SIGMAR1 (0.50) SIGMAR1ACHEBCHEUBE2MDCUN1D1
SCHEMBL8551176 0.77 PGR (0.54) MAPK1SIGMAR1ACHEKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US claimed
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed