SCHEMBL8551176

SCHEMBL8551176

Nc1cc([N+](=O)[O-])ccc1C(=O)OC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.54
CHRM2 P08172 1/20 0.54
ABCB1 P08183 1/20 0.54
HTR1A P08908 1/20 0.54
ADRA2A P08913 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CHRM1 P11229 1/20 0.54
DRD1 P21728 1/20 0.54
TBXA2R P21731 1/20 0.54
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
ADRA1A P35348 1/20 0.54
OPRM1 P35372 1/20 0.54
DRD3 P35462 1/20 0.54
SLC6A3 Q01959 1/20 0.54
KCNH2 Q12809 1/20 0.54
CACNA1C Q13936 1/20 0.54
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
SIGMAR1 Q99720 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553603 0.85 BCHE (0.54) ADRA2ASLC6A2ADRA1ADRD3SLC6A3
Hydrochloric Acid SCHEMBL8553924 0.84 BCHE (0.53) ADRA2ASLC6A2ADRA1ADRD3SLC6A3
SCHEMBL8552042 0.84 BCHE (0.53) SIGMAR1
SCHEMBL8550210 0.84 SLC6A12 (0.54) ADRA2ASLC6A2ADRA1ADRD3SLC6A3
SCHEMBL8551366 0.83 BCHE (0.52) ADRA2ASLC6A2ADRA1ADRD3SLC6A3
SCHEMBL8550767 0.83 BCHE (0.52) ADRA2ASLC6A2ADRA1ADRD3SLC6A3
Hydrochloric Acid SCHEMBL8554134 0.83 BCHE (0.52) SIGMAR1MEN1KMT2A
SCHEMBL8551172 0.83 BCHE (0.52) CHRM2DRD3SIGMAR1MAPTKMT2A
Hydrochloric Acid SCHEMBL8550148 0.83 SLC6A12 (0.53) ADRA2ASLC6A2ADRA1ADRD3SLC6A3
SCHEMBL8551099 0.83 MAPT (0.66) CHRM2ALDH1A1LMNASIGMAR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed