SCHEMBL8550870

SCHEMBL8550870

COC(=O)CCc1cc(N)ccc1OC

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
CYP19A1 P11511 1/20 0.43
PDE4D Q08499 1/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
RAD52 P43351 1/20 0.42
GFER P55789 1/20 0.42
TNF P01375 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1531406 0.88 GAA (0.57) TAAR1ALDH1A1GAAMAPTTSHR
SCHEMBL6350941 0.87 CYP4F2 (0.49) ADRA1ATAAR1ALDH1A1GAAMAPT
SCHEMBL11376820 0.86 ALDH1A1 (0.50) ADRA1ATAAR1ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL6976943 0.85 CYP4F2 (0.48) ADRA1ATAAR1ALDH1A1GAAMAPT
SCHEMBL9159002 0.84 HSD17B10 (0.49) ALDH1A1GAAMAPTTSHRMAPK1
SCHEMBL5034496 0.83 BACE1 (0.48) ALDH1A1PDE4D
SCHEMBL64208 0.83 MTNR1A (0.61) ADRA1ATAAR1MTNR1AMTNR1B
SCHEMBL2967999 0.82 ALDH1A1 (0.51) ALDH1A1MAPTTSHR
SCHEMBL8393174 0.82 GAA (0.43) ADRA1ATAAR1ALDH1A1GAAMAPT
SCHEMBL6157993 0.81 L3MBTL1 (0.43) ALDH1A1GAAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8318731-B2 Pyrrolopyrimidines JANSSEN PHARMACEUTICA NV (BE) 2012-11-27 US disclosed
US-8318731-B2 Pyrrolopyrimidines JANSSEN PHARMACEUTICA NV (BE) 2012-11-27 US disclosed
US-20100204197-A1 PYRROLOPYRIMIDINES JANSSEN PHARMACEUTICA NV (BE) 2010-08-12 US disclosed
US-20100204197-A1 PYRROLOPYRIMIDINES JANSSEN PHARMACEUTICA NV (BE) 2010-08-12 US disclosed
WO-1998018464-A1 SUBSTITUTED TRICYCLICS ELI LILLY AND COMPANY (US) 1998-05-07 WO disclosed
EP-0839806-A1 Substituted tricyclics ELI LILLY AND COMPANY (US) 1998-05-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100204197-A1 PYRROLOPYRIMIDINES PLK4, PLK2, PLK3 ADRA1A 3662/4885TAAR1 4222/4885ALDH1A1 2934/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.