SCHEMBL8550937

SCHEMBL8550937

CC(=O)c1c(F)cccc1N1CCN(CCc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
OPRM1 P35372 1/20 0.53
ADRA1D P25100 4/20 0.53
ADRA1A P35348 4/20 0.53
ADRA1B P35368 4/20 0.53
CYP2C9 P11712 1/20 0.50
HTR1A P08908 3/20 0.49
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692763 0.80 CYP1A2 (0.54) KMT2AMEN1ALDH1A1CYP2C9HTR1A
SCHEMBL8550916 0.78 MEN1 (0.55) KMT2AMEN1ALDH1A1ADRA1DADRA1A
SCHEMBL1537856 0.77 KDM4E (0.55) KMT2AALDH1A1CYP2C9DRD2
Ammonia Solution, Strong SCHEMBL27497850 0.76 KDM4E (0.54) KMT2AALDH1A1CYP2C9DRD2
SCHEMBL2905333 0.74 OPRM1 (0.52) KMT2AMEN1OPRM1HTR1ADRD2
SCHEMBL5364769 0.73 CYP1A2 (0.49) CYP2C9HTR1ADRD2HTR2AHTR2C
SCHEMBL11109442 0.73 HTR1A (0.63) KMT2AMEN1ALDH1A1ADRA1DADRA1A
Hydrochloric Acid SCHEMBL6017134 0.73 HTR1A (0.56) KMT2AMEN1ALDH1A1ADRA1DADRA1A
SCHEMBL2766780 0.72 ADRA1D (0.54) KMT2AMEN1ALDH1A1OPRM1ADRA1D
SCHEMBL2767637 0.72 HTR1A (0.54) KMT2AMEN1ALDH1A1ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed