SCHEMBL8551238

SCHEMBL8551238

Cc1oc2ccc(NC(=S)N3CCNCC3)cc2c1CCN(C)Cc1ccc2ccncc2c1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.37
EGFR P00533 1/20 0.34
LCK P06239 1/20 0.34
CSF1R P07333 1/20 0.34
KDR P35968 1/20 0.34
ERBB4 Q15303 1/20 0.34
MAPK14 Q16539 1/20 0.34
KDM4E B2RXH2 9/20 0.34
GAA P10253 9/20 0.34
MAPT P10636 7/20 0.34
RAD52 P43351 3/20 0.34
LMNA P02545 2/20 0.33
PRMT3 O60678 1/20 0.33
ALDH1A1 P00352 6/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RAB9A P51151 1/20 0.32
PHGDH O43175 1/20 0.32
ROCK2 O75116 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7145107 0.86 MAPT (0.43) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL8547927 0.85 ROCK1 (0.37) ROCK1EGFRLCKCSF1RKDR
SCHEMBL8548082 0.85 MKNK1 (0.38) EGFRLCKCSF1RKDRERBB4
SCHEMBL8550959 0.80 KDM4E (0.39) ROCK1KDM4EGAAMAPTRAD52
SCHEMBL8550329 0.80 KDM4E (0.40) ROCK1EGFRLCKCSF1RKDR
SCHEMBL8546411 0.78 ROCK2 (0.37) ROCK1EGFRLCKCSF1RKDR
SCHEMBL8550195 0.75 MEN1 (0.44) ROCK1KDM4EGAAMAPTALDH1A1
SCHEMBL8552082 0.72 KDM4E (0.45) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL8194168 0.70 TLR9 (0.43) SMN1; SMN2RAB9A
SCHEMBL8704913 0.70 MKNK1 (0.38) EGFRLCKCSF1RKDRERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed