SCHEMBL8551676

SCHEMBL8551676

CC(CCC(=O)CCC(C)(c1ccccc1)c1ccccc1)N(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.46
GRIN2A Q12879 6/20 0.46
GRIN2D O15399 5/20 0.46
GRIN2C Q14957 5/20 0.46
GRIN2B Q13224 4/20 0.46
OPRM1 P35372 2/20 0.46
KCNH2 Q12809 2/20 0.46
CACNA1F O60840 1/20 0.46
ABCB1 P08183 1/20 0.46
CYP2B6 P20813 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
CACNA1D Q01668 1/20 0.46
CACNA1S Q13698 1/20 0.46
CACNA1C Q13936 1/20 0.46
MRGPRX2 Q96LB1 1/20 0.46
CHRNB2 P17787 2/20 0.45
CHRNB4 P30926 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551678 0.74 HTR2A (0.47) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL20484039 0.73 CHRNB2 (0.49) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL75391 0.72 ALDH1A1 (0.72) OPRM1DRD4DRD3ALDH1A1ESR1
SCHEMBL2095353 0.70 CYP3A4 (0.53) KCNH2ALDH1A1ESR1CYP3A4ESR2
SCHEMBL27757219 0.69 GRIN1 (0.46) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL10439905 0.69 GRIN1 (0.52) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL8658460 0.68 GRIN1 (0.55) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL8698880 0.67 ALDH1A1 (0.50) ALDH1A1ESR1CYP3A4ESR2
SCHEMBL11140237 0.67 GRIN2D (0.41) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL11715175 0.66 CYP2C19 (0.59) OPRM1DRD3ALDH1A1ESR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827502-A1 METHADONE DERIVATIVES AND PROTEIN AND POLYPEPTIDE METHADONE DERIVATIVE CONJUGATES AND LABELS BIOSITE DIAGNOSTICS INC. (US) 1998-03-11 EP disclosed
WO-1996031496-A1 METHADONE DERIVATIVES AND PROTEIN AND POLYPEPTIDE METHADONE DERIVATIVE CONJUGATES AND LABELS BIOSITE DIAGNOSTICS, INCORPORATED (US) 1996-10-10 WO disclosed