SCHEMBL8551678

SCHEMBL8551678

CC(CCC(=O)CCCC(c1ccccc1)c1ccccc1)N(C)C

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.47
HRH1 P35367 4/20 0.47
CHRNB2 P17787 5/20 0.47
CHRNB4 P30926 5/20 0.47
CHRNA4 P43681 5/20 0.47
CHRNA3 P32297 4/20 0.47
SIGMAR1 Q99720 2/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
TBXAS1 P24557 1/20 0.40
GRM2 Q14416 1/20 0.39
GRM3 Q14832 1/20 0.39
CASR P41180 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20484039 0.84 CHRNB2 (0.49) HTR2AHRH1CHRNB2CHRNB4CHRNA4
SCHEMBL8494372 0.83 HRH1 (0.54) HTR2AHRH1SIGMAR1MTNR1AMTNR1B
SCHEMBL27593431 0.77 SIGMAR1 (0.49) HTR2AHRH1SIGMAR1MTNR1AMTNR1B
SCHEMBL8494351 0.76 MTNR1A (0.52) HTR2AHRH1MTNR1AMTNR1BTBXAS1
SCHEMBL5402685 0.74 TBXAS1 (0.49) HTR2AHRH1MTNR1AMTNR1BTBXAS1
SCHEMBL8551676 0.74 GRIN1 (0.46) CHRNB2CHRNB4CHRNA4CHRNA3
SCHEMBL31108377 0.73 ASAH1 (0.52) SIGMAR1TBXAS1
SCHEMBL7011219 0.73 ASAH1 (0.52) SIGMAR1TBXAS1
SCHEMBL3943859 0.73 MTNR1A (0.47) HTR2AHRH1SIGMAR1MTNR1AMTNR1B
SCHEMBL5692956 0.73 TBXAS1 (0.63) HTR2AHRH1MTNR1AMTNR1BTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827502-A1 METHADONE DERIVATIVES AND PROTEIN AND POLYPEPTIDE METHADONE DERIVATIVE CONJUGATES AND LABELS BIOSITE DIAGNOSTICS INC. (US) 1998-03-11 EP disclosed
WO-1996031496-A1 METHADONE DERIVATIVES AND PROTEIN AND POLYPEPTIDE METHADONE DERIVATIVE CONJUGATES AND LABELS BIOSITE DIAGNOSTICS, INCORPORATED (US) 1996-10-10 WO disclosed