SCHEMBL8548542

SCHEMBL8548542

Cc1ccc(-c2n[nH]c(=O)c3c(C(F)(F)F)cccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.47
NAMPT P43490 2/20 0.47
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PARP1 P09874 2/20 0.43
ATM Q13315 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
AR P10275 1/20 0.41
ENPP1 P22413 1/20 0.40
LMNA P02545 2/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
MAPT P10636 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551845 0.88 ROCK2 (0.48) ROCK2NAMPTALDH1A1KMT2ASMN1; SMN2
SCHEMBL8551517 0.87 NPSR1 (0.57) ROCK2NAMPTALDH1A1MEN1KMT2A
SCHEMBL8547192 0.79 ALDH1A1 (0.48) ROCK2ALDH1A1MAPK1MEN1KMT2A
SCHEMBL3707918 0.77 ROCK2 (0.57) ROCK2NAMPTALDH1A1MAPK1PARP1
SCHEMBL8551923 0.77 ALDH1A1 (0.43) ROCK2NAMPTALDH1A1MAPK1SMN1; SMN2
SCHEMBL8549961 0.76 MEN1 (0.44) ALDH1A1MAPK1MEN1KMT2ASMN1; SMN2
SCHEMBL8552718 0.75 ALDH1A1 (0.42) ALDH1A1MAPK1MEN1KMT2ASMN1; SMN2
SCHEMBL8547799 0.75 KMT2A (0.43) ALDH1A1MAPK1MEN1KMT2ASMN1; SMN2
SCHEMBL1786578 0.75 ATM (0.73) ROCK2ALDH1A1MAPK1MEN1KMT2A
SCHEMBL30602968 0.74 PIK3CA (0.46) ROCK2NAMPTMAPK1PARP1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed