SCHEMBL8553958

SCHEMBL8553958

O=C(O)CN1CCC(CNC(=O)c2nnc(C3CCNCC3)s2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.42
HTR4 Q13639 1/20 0.38
EP300 Q09472 1/20 0.38
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
KCNH2 Q12809 1/20 0.35
CACNA1I Q9P0X4 1/20 0.35
PLAT P00750 1/20 0.35
EIF4E P06730 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552049 0.85 SMYD3 (0.43)
Bromide SCHEMBL8554036 0.80 GSK3B (0.42) GSK3BHTR4EP300
SCHEMBL8553962 0.77 ITGB3 (0.34) PLAT
SCHEMBL8555209 0.77 KDM4E (0.36) PLAT
SCHEMBL8552893 0.74 SMYD3 (0.43)
Hydrochloric Acid SCHEMBL8551719 0.73 SMYD3 (0.42)
SCHEMBL8625016 0.72 KDM4E (0.49) HTR4
Hydrochloric Acid SCHEMBL8552279 0.71 MEN1 (0.38) HTR4EIF4EMKNK1MKNK2
Hydrochloric Acid SCHEMBL8549592 0.70 GSK3B (0.40) GSK3BHTR4EP300KCNH2CACNA1I
SCHEMBL8550362 0.70 SMYD3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed