SCHEMBL8552247

SCHEMBL8552247

CS(=O)(=O)OC(C(=O)c1ccccc1)C1CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
SLC6A4 P31645 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.35
CCR8 P51685 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CACNA2D1 P54289 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNB1 Q02641 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27512854 0.80 CYP3A4 (0.42) OPRD1ALDH1A1CYP3A4SLC6A4SLC6A2
SCHEMBL4047557 0.75 ALDH1A1 (0.38) ALDH1A1CYP3A4
SCHEMBL4047562 0.75 ALDH1A1 (0.38) ALDH1A1CYP3A4
SCHEMBL27585299 0.73 LMNA (0.46) OPRD1ALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL27486159 0.73 OPRD1 (0.44) OPRD1ALDH1A1SLC6A4SLC6A3SMYD3
SCHEMBL29277061 0.73 OPRD1 (0.44) OPRD1ALDH1A1SLC6A4SLC6A3CCR8
SCHEMBL27269213 0.73 SLC6A4 (0.42) OPRD1SLC6A4SLC6A2SLC6A3SIGMAR1
SCHEMBL10712783 0.71 ALDH1A1 (0.51) ALDH1A1CYP3A4
SCHEMBL7232624 0.71 OPRD1 (0.48) OPRD1SLC6A4SLC6A2SLC6A3SMYD3
SCHEMBL458925 0.70 CPN1 (0.34) ALDH1A1CYP3A4MMP1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed