SCHEMBL8552317

SCHEMBL8552317

Cc1sc2ccc(NC(=O)c3ccoc3)cc2c1CCNCc1nnco1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.36
KCNK3 O14649 1/20 0.35
KCNK9 Q9NPC2 1/20 0.35
MAPK14 Q16539 6/20 0.34
HSPB1 P04792 1/20 0.34
EGFR P00533 1/20 0.33
LCK P06239 1/20 0.33
LRRK2 Q5S007 4/20 0.32
TRPV1 Q8NER1 4/20 0.32
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 2/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
RECQL P46063 1/20 0.31
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547929 0.84 MAPK14 (0.36) RAB9AKCNK3KCNK9MAPK14HSPB1
SCHEMBL7138889 0.83 HTR1F (0.45) RAB9AKCNK3KCNK9LRRK2MEN1
SCHEMBL8548429 0.69 LRRK2 (0.36) RAB9AKCNK3KCNK9MAPK14HSPB1
SCHEMBL7145099 0.69 HTR1F (0.51) RAB9AKCNK3KCNK9MAPK14HSPB1
SCHEMBL8553318 0.64 MAPT (0.43) RAB9AMEN1MAPTKMT2AKDM4E
SCHEMBL13546243 0.62 KCNK3 (0.60) RAB9AKCNK3KCNK9MAPK14HSPB1
SCHEMBL8546818 0.62 DYRK1A (0.36) RAB9AEGFRMEN1MAPTKMT2A
SCHEMBL18027799 0.60 RAB9A (0.65) RAB9AKCNK3KCNK9MEN1MAPT
SCHEMBL7142217 0.60 HTR1F (0.62) RAB9ALRRK2MEN1MAPTKMT2A
SCHEMBL8288209 0.59 HDAC1 (0.69) RAB9AKCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed