SCHEMBL8548429

SCHEMBL8548429

Cc1oc2ccc(NC(=O)c3ccoc3)cc2c1CCN(C)Cc1nnco1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.36
MAPK14 Q16539 6/20 0.35
HSPB1 P04792 1/20 0.35
RAB9A P51151 1/20 0.35
KCNK3 O14649 1/20 0.35
KCNK9 Q9NPC2 1/20 0.35
HTR1F P30939 2/20 0.35
CA9 Q16790 1/20 0.33
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32
SNCA P37840 2/20 0.32
EGFR P00533 1/20 0.32
LCK P06239 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547929 0.85 MAPK14 (0.36) LRRK2MAPK14HSPB1RAB9AKCNK3
SCHEMBL7145099 0.85 HTR1F (0.51) LRRK2MAPK14HSPB1RAB9AKCNK3
SCHEMBL8549783 0.71 GRM5 (0.37) RAB9AHTR1FCA9
SCHEMBL8549636 0.71 HTR1F (0.51) RAB9AKCNK3KCNK9HTR1FCA9
SCHEMBL8548549 0.71 HTR1F (0.50) MAPK14RAB9AKCNK3KCNK9HTR1F
SCHEMBL8552317 0.69 RAB9A (0.36) LRRK2MAPK14HSPB1RAB9AKCNK3
SCHEMBL7138889 0.69 HTR1F (0.45) LRRK2RAB9AKCNK3KCNK9HTR1F
SCHEMBL8552580 0.69 HTR1F (0.65) RAB9AKCNK3KCNK9HTR1FSNCA
SCHEMBL8547488 0.69 HTR1F (0.53) RAB9AKCNK3HTR1FCA9SNCA
SCHEMBL8548295 0.68 RAB9A (0.51) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed