SCHEMBL8552369

SCHEMBL8552369

CC(CC(Oc1cccc(-c2ccccc2)c1)c1cccnc1)OC(=O)C(=O)OC(C)CC(Oc1cccc(-c2ccccc2)c1)c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.45
KCNA5 P22460 4/20 0.43
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
DGAT2 Q96PD7 2/20 0.41
CTSA P10619 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
PTAFR P25105 1/20 0.39
KCNH2 Q12809 1/20 0.39
HTT P42858 1/20 0.39
FFAR1 O14842 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
SUCNR1 Q9BXA5 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554522 0.87 KCNA5 (0.42) KCNA5CTSLCTSSCTSKFFAR1
SCHEMBL8550969 0.86 EPHX1 (0.46) EPHX1KCNA5CTSLCTSSCTSK
SCHEMBL8553452 0.85 SUCNR1 (0.41) HTTADRB1ADRB3AKR1C3AKR1C2
SCHEMBL8549826 0.84 KCNA5 (0.43) KCNA5CTSLCTSSCTSKKCNH2
SCHEMBL8551344 0.84 CYP19A1 (0.47) PTAFRSUCNR1
SCHEMBL8556196 0.83 PDE4D (0.41) AKR1C3AKR1C2
SCHEMBL8553713 0.82 CYP17A1 (0.42) CTSLCTSSCTSKADRB1ADRB3
SCHEMBL8554677 0.77 EPHX1 (0.42) EPHX1KCNA5CTSLCTSSCTSK
SCHEMBL2526 0.76 HTT (0.44) KCNA5HTT
SCHEMBL8118689 0.76 KCNA5 (0.48) KCNA5DGAT2PTAFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed