SCHEMBL8553713

SCHEMBL8553713

CNS(=O)(=O)c1cccc(-c2ccc(OC(CC(C)OC(=O)C(=O)OC(C)CC(Oc3ccc(-c4cccc(S(=O)(=O)NC)c4)cc3)c3cccnc3)c3cccnc3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.42
CYP3A4 P08684 1/20 0.42
LARS1 Q9P2J5 3/20 0.41
MAPT P10636 1/20 0.41
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
F10 P00742 1/20 0.37
F7 P08709 1/20 0.37
F3 P13726 1/20 0.37
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
ADAMTS4 O75173 1/20 0.37
TBXAS1 P24557 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554522 0.83 KCNA5 (0.42) MAPTPSEN1PSEN2APH1BNCSTN
SCHEMBL8551344 0.83 CYP19A1 (0.47) CYP11B1CYP11B2
SCHEMBL8552369 0.82 EPHX1 (0.45) CTSLCTSSCTSKADRB1ADRB3
SCHEMBL8549826 0.81 KCNA5 (0.43) CYP17A1CYP11B1CYP11B2PSEN1PSEN2
SCHEMBL8556196 0.80 PDE4D (0.41) MAPTCYP11B1CYP11B2LMNA
SCHEMBL8553452 0.74 SUCNR1 (0.41) MAPTADRB1ADRB3LMNA
SCHEMBL7966525 0.73 PTAFR (0.44) CYP17A1CYP3A4LARS1MAPTCYP11B1
SCHEMBL7966529 0.73 PTAFR (0.44) CYP17A1CYP3A4LARS1MAPTCYP11B1
SCHEMBL8481898 0.73 ADAMTS4 (0.44) CYP17A1CYP3A4MAPTCYP11B1CYP11B2
SCHEMBL8118375 0.73 KCNA5 (0.49) CYP3A4MAPTADRB1ADRB3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed