SCHEMBL8554677

SCHEMBL8554677

CC(=O)Oc1cccc(-c2ccc(OC(CC(C)O)c3cccnc3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
ADRB3 P13945 3/20 0.40
ADRB1 P08588 2/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 2/20 0.40
GAA P10253 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
DGAT2 Q96PD7 4/20 0.40
PTAFR P25105 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
KCNA5 P22460 1/20 0.39
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8118689 0.88 KCNA5 (0.48) SMN1; SMN2NPC1TP53RAB9AMAPT
SCHEMBL8550969 0.87 EPHX1 (0.46) EPHX1SMN1; SMN2ADRB3ADRB1RXRA
SCHEMBL8555638 0.87 SUCNR1 (0.43) ADRB3ADRB1LMNAGAAPTAFR
SCHEMBL8551743 0.85 KMO (0.51) ADRB3ADRB1LMNAGAARXRA
SCHEMBL8552914 0.84 CYP17A1 (0.48) PKMLMNA
SCHEMBL8552459 0.84 CYP17A1 (0.44) ADRB3ADRB1PTAFRFFAR1
SCHEMBL8552624 0.84 CYP19A1 (0.47) SMN1; SMN2ADRB3ADRB1MKNK1MKNK2
SCHEMBL8109544 0.84 SMN1; SMN2 (0.44) SMN1; SMN2PKMADRB3ADRB1GAA
SCHEMBL8118264 0.83 DGAT2 (0.39) ADRB3ADRB1DGAT2KCNA5FFAR1
SCHEMBL8118468 0.83 KCNA5 (0.45) ADRB3ADRB1KCNA5FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed