SCHEMBL8552459

SCHEMBL8552459

CC(O)CC(Oc1ccc(-c2cccc(O)c2)cc1)c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 6/20 0.44
CYP19A1 P11511 5/20 0.40
CYP11B1 P15538 4/20 0.40
CYP11B2 P19099 4/20 0.40
CYP3A4 P08684 5/20 0.40
HSD17B1 P14061 3/20 0.39
HSD17B2 P37059 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2B6 P20813 1/20 0.39
FFAR1 O14842 1/20 0.39
PTAFR P25105 1/20 0.38
ADRB3 P13945 3/20 0.37
ADRB1 P08588 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552624 0.88 CYP19A1 (0.47) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8109544 0.88 SMN1; SMN2 (0.44) CYP17A1CYP19A1CYP3A4CYP2C9CYP2D6
SCHEMBL8123208 0.88 MKNK1 (0.46) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8118689 0.88 KCNA5 (0.48) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8118264 0.88 DGAT2 (0.39) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8118468 0.88 KCNA5 (0.45) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8552479 0.87 PRKCI (0.44) CYP17A1CYP19A1CYP11B1CYP11B2FFAR1
SCHEMBL8551523 0.86 CYP17A1 (0.47) CYP17A1CYP19A1CYP3A4
SCHEMBL8117772 0.85 KCNA5 (0.45) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8672155 0.85 KCNA5 (0.48) CYP17A1CYP11B1CYP11B2CYP3A4FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed