SCHEMBL8551523

SCHEMBL8551523

CC(O)CC(Oc1ccc(O)cc1)c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 1/20 0.38
GAA P10253 2/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
RECQL P46063 1/20 0.38
HSD17B10 Q99714 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.37
HTT P42858 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP3A5 P20815 2/20 0.36
GRIN1 Q05586 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7772046 0.88 SLC6A4 (0.42) SMN1; SMN2LMNAL3MBTL1SLC6A2SLC6A4
SCHEMBL7773934 0.88 SLC6A4 (0.42) SMN1; SMN2LMNAL3MBTL1SLC6A2SLC6A4
SCHEMBL8552624 0.87 CYP19A1 (0.47) CYP17A1SMN1; SMN2ALDH1A1CYP3A4CYP19A1
SCHEMBL8109544 0.87 SMN1; SMN2 (0.44) CYP17A1SMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL8552459 0.86 CYP17A1 (0.44) CYP17A1CYP3A4CYP19A1
SCHEMBL8551073 0.85 MAPK1 (0.47) SMN1; SMN2LMNAL3MBTL1SLC6A2SLC6A3
SCHEMBL8133883 0.85 CYP17A1 (0.40) CYP17A1SMN1; SMN2LMNAL3MBTL1SLC6A2
SCHEMBL8551928 0.84 CYP11B1 (0.43) SMN1; SMN2LMNAALDH1A1ALOX15HSD17B10
SCHEMBL8550686 0.82 KCNA5 (0.43) CYP17A1SLC6A4CYP3A4CYP3A5CYP19A1
SCHEMBL8550029 0.82 CYP19A1 (0.47) CYP17A1ALDH1A1HPGDCYP3A4CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed