SCHEMBL8672155

SCHEMBL8672155

CC(O)CC(Oc1ccc(-c2cccc(C(F)(F)F)c2)cc1)c1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 4/20 0.48
FFAR1 O14842 2/20 0.47
CYP3A4 P08684 2/20 0.45
CYP3A5 P20815 1/20 0.45
KCNH2 Q12809 1/20 0.45
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
NPY5R Q15761 1/20 0.39
ADAMTS4 O75173 1/20 0.38
MMP13 P45452 1/20 0.38
GRIN1 Q05586 4/20 0.38
GRIN2B Q13224 4/20 0.38
PNMT P11086 1/20 0.38
CYP17A1 P05093 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8118264 0.86 DGAT2 (0.39) KCNA5FFAR1CYP3A4KCNH2CYP17A1
SCHEMBL8552459 0.85 CYP17A1 (0.44) FFAR1CYP3A4CYP17A1CYP11B1CYP11B2
SCHEMBL8109544 0.85 SMN1; SMN2 (0.44) KCNA5CYP3A4KCNH2GAACYP17A1
SCHEMBL8552624 0.85 CYP19A1 (0.47) KCNA5CYP3A4ALDH1A1CYP17A1CYP11B1
SCHEMBL8118689 0.84 KCNA5 (0.48) KCNA5CYP3A4NPY5RCYP17A1CYP11B1
SCHEMBL8123208 0.84 MKNK1 (0.46) FFAR1CYP3A4CYP17A1CYP11B1CYP11B2
SCHEMBL8118468 0.84 KCNA5 (0.45) KCNA5FFAR1CYP3A4CYP3A5CYP17A1
SCHEMBL8552479 0.83 PRKCI (0.44) FFAR1CYP17A1CYP11B1CYP11B2
SCHEMBL8117772 0.82 KCNA5 (0.45) KCNA5CYP3A4KCNH2ALDH1A1CYP17A1
SCHEMBL8555638 0.82 SUCNR1 (0.43) KCNA5FFAR1KCNH2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed