SCHEMBL8552621

SCHEMBL8552621

CS(=O)(=O)c1ccc(-c2[nH]c(-c3ccc(Cl)cc3)nc2CCl)cc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.55
PTGS1 P23219 5/20 0.55
MAPK14 Q16539 2/20 0.47
ALDH1A1 P00352 1/20 0.47
ALOX5 P09917 1/20 0.47
CSNK1A1 P48729 1/20 0.47
CSNK1D P48730 1/20 0.47
CSNK1E P49674 1/20 0.47
MAPK11 Q15759 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CSNK1A1L Q8N752 1/20 0.47
SCD O00767 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796825 0.88 PTGS2 (0.54) PTGS2PTGS1MAPK14ALDH1A1ALOX5
SCHEMBL8556092 0.85 PTGS2 (0.51) PTGS2PTGS1MAPK14ALDH1A1ALOX5
SCHEMBL5597068 0.82 PTGS1 (0.75) PTGS2PTGS1MAPK14ALDH1A1ALOX5
SCHEMBL19350071 0.82 CTSS (0.46) PTGS2PTGS1MAPK14ALDH1A1ALOX5
SCHEMBL3246495 0.81 PTGS2 (0.50) PTGS2PTGS1SCD
SCHEMBL19350079 0.75 MAPK1 (0.49) MAPK14ALDH1A1MAPK11SMN1; SMN2
Hydrochloric Acid SCHEMBL8963881 0.74 MAPK1 (0.47) MAPK14ALDH1A1MAPK11SMN1; SMN2
Hydrochloric Acid SCHEMBL8963707 0.74 MAPK13 (0.44) MAPK14ALDH1A1MAPK11SMN1; SMN2
SCHEMBL15245084 0.72 SCD (0.65) PTGS2SCD
SCHEMBL7088050 0.72 PTGS1 (0.66) PTGS2PTGS1MAPK14ALDH1A1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880504-A1 HETEROCYCLO-SUBSTITUTED IMIDAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-12-02 EP disclosed
WO-1997027181-A1 HETEROCYCLO-SUBSTITUTED IMIDAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-07-31 WO disclosed