SCHEMBL8552847

SCHEMBL8552847

Cc1ccc(O)c2c1NC(=O)C2(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
CNR1 P21554 1/20 0.41
GPR35 Q9HC97 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
PDK2 Q15119 4/20 0.39
PDK4 Q16654 3/20 0.38
PDK1 Q15118 1/20 0.38
PDK3 Q15120 1/20 0.38
KMT2A Q03164 4/20 0.36
MEN1 O00255 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
DAO P14920 3/20 0.34
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
XBP1 P17861 1/20 0.33
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556238 0.76 PDK2 (0.34) ALDH1A1HTTCNR1GPR35GPR55
SCHEMBL8556960 0.75 PDK2 (0.44) CNR1PDK2PDK4PDK1PDK3
SCHEMBL9095539 0.74 ALDH1A1 (0.36) ALDH1A1HTTCNR1GPR35GPR55
SCHEMBL8557438 0.73 PDK2 (0.42) HTTPDK2KMT2AMEN1MAPT
SCHEMBL8559099 0.72 TYR (0.44) HTTPDK2KMT2AMEN1MAPT
SCHEMBL9094130 0.70 ALDH1A1 (0.36) ALDH1A1HTTCNR1GPR35GPR55
SCHEMBL8559248 0.70 ALDH1A1 (0.42) ALDH1A1HTTCNR1GPR35GPR55
SCHEMBL2264510 0.69 PDK2 (0.62) HTTCNR1GPR35GPR55PDK2
SCHEMBL3150359 0.69 PDK2 (0.52) ALDH1A1PDK2PDK4PDK1PDK3
SCHEMBL8554583 0.69 PDE4B (0.37) ALDH1A1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653426-B1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA CO (JP) 1998-07-22 EP disclosed
US-5510366-A INOTROPIC, ANTIARRHYMTHMIA AGENTS, VASODILATORS KOWA CO., LTD. (JP) 1996-04-23 US disclosed
EP-0653426-A1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA COMPANY, LTD. (JP) 1995-05-17 EP disclosed