SCHEMBL8557438

SCHEMBL8557438

CCCCc1ccc(O)c2c1NC(=O)C2(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.42
TYR P14679 3/20 0.41
ELANE P08246 3/20 0.40
CTSG P08311 3/20 0.40
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX5 P09917 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
CTRC Q99895 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559099 0.96 TYR (0.44) PDK2TYRELANECTSGMEN1
SCHEMBL8557956 0.94 TYR (0.47) PDK2TYRELANECTSGMEN1
SCHEMBL8556960 0.91 PDK2 (0.44) PDK2TYRELANECTSGALOX5
SCHEMBL8552847 0.73 ALDH1A1 (0.41) PDK2ELANECTSGMEN1MAPT
SCHEMBL8554202 0.72 MEN1 (0.35) PDK2TYRELANECTSGMEN1
SCHEMBL8557800 0.71 KDM4E (0.35) PDK2ELANEMEN1CYP3A4ALOX5
SCHEMBL8557767 0.70 THRA (0.36) PDK2ELANEMEN1MAPTTSHR
SCHEMBL8598630 0.69 MEN1 (0.34) PDK2ELANECTSGMEN1ALOX5
SCHEMBL2382145 0.64 TYR (0.61) TYRELANECTSGMEN1TP53
SCHEMBL167918 0.63 TYR (0.55) TYRELANECTSGMEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653426-B1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA CO (JP) 1998-07-22 EP disclosed
US-5510366-A INOTROPIC, ANTIARRHYMTHMIA AGENTS, VASODILATORS KOWA CO., LTD. (JP) 1996-04-23 US disclosed
EP-0653426-A1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA COMPANY, LTD. (JP) 1995-05-17 EP disclosed