SCHEMBL8552960

SCHEMBL8552960

CC(O)CC(Oc1ccc(-c2ccc(Cl)cc2Cl)cc1)c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARS1 P56192 5/20 0.41
DAGLA Q9Y4D2 2/20 0.40
CYP3A4 P08684 3/20 0.39
CYP3A5 P20815 2/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
PDK1 Q15118 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 1/20 0.38
MME P08473 1/20 0.38
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CYP19A1 P11511 1/20 0.36
SLC6A2 P23975 1/20 0.36
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555184 0.88 KCNA5 (0.40) CYP3A4PDK1SLC6A4SMN1; SMN2CYP17A1
SCHEMBL8118468 0.86 KCNA5 (0.45) CYP3A4CYP3A5SLC6A4SLC6A3CYP19A1
SCHEMBL8550686 0.86 KCNA5 (0.43) CYP3A4CYP3A5SLC6A4CYP19A1CYP17A1
SCHEMBL8117056 0.84 CYP3A4 (0.40) CYP3A4CYP3A5LMNAMMEMEN1
SCHEMBL8552624 0.82 CYP19A1 (0.47) CYP3A4SMN1; SMN2CYP19A1CYP17A1CYP11B1
SCHEMBL8109544 0.82 SMN1; SMN2 (0.44) CYP3A4SLC6A4SLC6A3HTTSMN1; SMN2
SCHEMBL8555652 0.81 PPARG (0.41) CYP3A4MMESMN1; SMN2NPSR1CYP17A1
SCHEMBL8133883 0.80 CYP17A1 (0.40) CYP3A4LMNAHPGDSLC6A4SLC6A3
SCHEMBL8551523 0.79 CYP17A1 (0.47) CYP3A4CYP3A5LMNAHPGDSLC6A4
SCHEMBL8552479 0.79 PRKCI (0.44) HPGDHTTSMN1; SMN2CYP19A1CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed