SCHEMBL8555652

SCHEMBL8555652

CC(O)CC(Oc1ccc(-c2ccccc2F)cc1)c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
KCNA5 P22460 3/20 0.41
KCNH2 Q12809 2/20 0.41
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
ALOX5AP P20292 2/20 0.37
FEN1 P39748 2/20 0.37
ROCK1 Q13464 2/20 0.37
PRKACA P17612 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
PRKX P51817 1/20 0.37
PRKCQ Q04759 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
ROCK2 O75116 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109544 0.86 SMN1; SMN2 (0.44) KCNA5KCNH2SMN1; SMN2CYP3A4CYP2C9
SCHEMBL8552624 0.83 CYP19A1 (0.47) KCNA5SMN1; SMN2CYP3A4CYP2C9CYP17A1
SCHEMBL8139574 0.83 ALOX5AP (0.39) KCNA5KCNH2ALOX5APFEN1SMN1; SMN2
SCHEMBL8117056 0.82 CYP3A4 (0.40) KCNA5AKR1C3AKR1C2CYP3A4MME
SCHEMBL8133883 0.81 CYP17A1 (0.40) KCNA5SMN1; SMN2CYP3A4CYP2C9CYP17A1
SCHEMBL8118264 0.81 DGAT2 (0.39) KCNA5KCNH2AKR1C3AKR1C2CYP3A4
SCHEMBL8551523 0.81 CYP17A1 (0.47) SMN1; SMN2CYP3A4CYP17A1GAA
SCHEMBL8552960 0.81 MARS1 (0.41) SMN1; SMN2CYP3A4NPSR1MMECYP17A1
SCHEMBL8119038 0.80 CYP11B1 (0.43) CYP3A4CYP11B1CYP11B2
SCHEMBL7772046 0.80 SLC6A4 (0.42) KCNA5SMN1; SMN2CYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed