SCHEMBL8550686

SCHEMBL8550686

CC(O)CC(Oc1ccc(-c2cc(Cl)cc(Cl)c2)cc1)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 6/20 0.43
KCND3 Q9UK17 1/20 0.43
SLC6A4 P31645 1/20 0.39
CYP3A4 P08684 3/20 0.39
CYP3A5 P20815 2/20 0.39
CYP17A1 P05093 2/20 0.38
ADRB3 P13945 4/20 0.36
ADRB1 P08588 3/20 0.36
SUCNR1 Q9BXA5 2/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CTSA P10619 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8118468 0.91 KCNA5 (0.45) KCNA5KCND3SLC6A4CYP3A4CYP3A5
SCHEMBL8117056 0.87 CYP3A4 (0.40) KCNA5KCND3CYP3A4CYP3A5CYP17A1
SCHEMBL8552624 0.87 CYP19A1 (0.47) KCNA5CYP3A4CYP17A1ADRB3ADRB1
SCHEMBL8109544 0.87 SMN1; SMN2 (0.44) KCNA5SLC6A4CYP3A4CYP17A1ADRB3
SCHEMBL8552960 0.86 MARS1 (0.41) SLC6A4CYP3A4CYP3A5CYP17A1CYP19A1
SCHEMBL8133883 0.85 CYP17A1 (0.40) KCNA5SLC6A4CYP3A4CYP17A1ADRB3
SCHEMBL8124227 0.84 CYP19A1 (0.39) KCNA5CYP3A4CYP17A1ADRB3ADRB1
SCHEMBL8552459 0.83 CYP17A1 (0.44) CYP3A4CYP17A1ADRB3ADRB1CYP19A1
SCHEMBL8118689 0.82 KCNA5 (0.48) KCNA5CYP3A4CYP17A1CYP19A1CYP11B1
SCHEMBL8118264 0.82 DGAT2 (0.39) KCNA5CYP3A4CYP17A1ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed