SCHEMBL8553015

SCHEMBL8553015

O=C(NNC1CCOCC1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
KMT2A Q03164 2/20 0.47
POLB P06746 2/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
PTGS2 P35354 1/20 0.46
CCR2 P41597 1/20 0.45
NAMPT P43490 1/20 0.45
KDM1A O60341 1/20 0.45
HPGD P15428 1/20 0.44
MEN1 O00255 1/20 0.44
KDM4E B2RXH2 1/20 0.43
KAT2B Q92831 1/20 0.43
BAZ2B Q9UIF8 1/20 0.43
HDAC3 O15379 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29268969 0.87 NPC1 (0.55) SMN1; SMN2KMT2APOLBMAPTNPC1
SCHEMBL364174 0.84 NPC1 (0.62) SMN1; SMN2KMT2ANPC1RAB9ANAMPT
SCHEMBL8180075 0.84 NPC1 (0.60) SMN1; SMN2KMT2APOLBMAPTNPC1
Water SCHEMBL30838095 0.83 NPC1 (0.60) SMN1; SMN2KMT2ANPC1RAB9ANAMPT
SCHEMBL6639389 0.82 RAB9A (0.61) SMN1; SMN2NPC1RAB9ACTDSP1PTGS2
SCHEMBL854076 0.81 NAMPT (0.49) NPC1RAB9ACTDSP1PTGS2NAMPT
SCHEMBL633936 0.78 NAMPT (0.61) SMN1; SMN2KMT2ANPC1RAB9ANAMPT
SCHEMBL29167802 0.78 NAMPT (0.61) SMN1; SMN2KMT2ANPC1RAB9ANAMPT
SCHEMBL13868569 0.78 NAMPT (0.61) SMN1; SMN2KMT2ANPC1RAB9ANAMPT
SCHEMBL10557090 0.77 CARM1 (0.52) KMT2ANPC1RAB9AMEN1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN claimed
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed
US-11253515-B2 Pharmaceutical compositions and dosage forms IGNYTA, INC. (US) 2022-02-22 US disclosed
US-20200163892-A1 PHARMACEUTICAL COMPOSITIONS AND DOSAGE FORMS IGNYTA, INC. (US) 2020-05-28 US disclosed
EP-3227276-A1 COMBINATIONS FOR THE TREATMENT OF NEUROBLASTOMA Ignyta, Inc. (US) 2017-10-11 EP disclosed
US-20170007599-A1 METHODS FOR TREATING NEUROBLASTOMA IGNYTA, INC. 2017-01-12 US disclosed
EP-3107541-A1 COMPOUNDS FOR TREATING PATIENTS WITH ROS1 MUTANT CANCER CELLS Ignyta, Inc. (US) 2016-12-28 EP disclosed
WO-2016089760-A1 COMBINATIONS FOR THE TREATMENT OF NEUROBLASTOMA IGNYTA, INC. (US) 2016-06-09 WO disclosed
WO-2015124697-A1 COMPOUNDS FOR TREATING PATIENTS WITH ROS1 MUTANT CANCER CELLS IGNYTA, INC. (US) 2015-08-27 WO disclosed
EP-0885890-A1 SULFONYLUREIDOPYRAZOLE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-12-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170007599-A1 METHODS FOR TREATING NEUROBLASTOMA NEK2, CSNK1G3, AHNAK SMN1; SMN2 58/4885KMT2A 802/4885POLB 2806/4885
US-20200163892-A1 PHARMACEUTICAL COMPOSITIONS AND DOSAGE FORMS CYP3A5, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, PAICS SMN1; SMN2 633/4885KMT2A 604/4885POLB 2988/4885
US-11253515-B2 Pharmaceutical compositions and dosage forms CYP3A5, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, PAICS SMN1; SMN2 633/4885KMT2A 604/4885POLB 2988/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.