SCHEMBL8553016

SCHEMBL8553016

O=c1[nH]nc(-c2ccc(Cl)cc2)c2cccc(Br)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.45
ATM Q13315 1/20 0.45
PDPK1 O15530 1/20 0.41
LMNA P02545 1/20 0.40
ROCK1 Q13464 3/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TNKS O95271 3/20 0.38
TNKS2 Q9H2K2 3/20 0.38
PARP2 Q9UGN5 2/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 2/20 0.38
GUSB P08236 1/20 0.38
POLB P06746 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548460 0.86 NPSR1 (0.62) NPSR1ATMROCK1KDM4EALDH1A1
SCHEMBL8552572 0.85 ALDH1A1 (0.48) NPSR1ATMROCK1KDM4EALDH1A1
SCHEMBL8552195 0.80 AR (0.42) NPSR1ATMPDPK1LMNAROCK1
SCHEMBL31014288 0.78 ATM (0.73) NPSR1ATMLMNAROCK1KDM4E
SCHEMBL706420 0.78 ATM (0.73) NPSR1ATMLMNAROCK1KDM4E
SCHEMBL8550946 0.77 ADORA2A (0.41) NPSR1ATMKDM4EALDH1A1MAPT
SCHEMBL8547990 0.77 NPSR1 (0.50) NPSR1ATMPDPK1LMNAROCK1
SCHEMBL8551285 0.74 AR (0.42) NPSR1ATMPDPK1LMNAROCK1
SCHEMBL8551565 0.74 KMT2A (0.42) NPSR1LMNAKDM4EALDH1A1MEN1
SCHEMBL8551583 0.74 NPSR1 (0.62) NPSR1ATMROCK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed