SCHEMBL8553115

SCHEMBL8553115

COC(=O)Oc1ccc2[nH]cc(C3=CCN(CCCCc4c[nH]c5ccc(C(=O)OC)cc45)CC3)c2c1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.59
KDM4E B2RXH2 1/20 0.59
ALOX15 P16050 1/20 0.59
APEX1 P27695 1/20 0.59
KMT2A Q03164 1/20 0.59
HSD17B10 Q99714 1/20 0.59
HTR1A P08908 3/20 0.58
DRD2 P14416 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
DRD4 P21917 1/20 0.50
CYP2C19 P33261 1/20 0.50
DRD3 P35462 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555961 0.93 HTR1A (0.68) TDP1KDM4EALOX15APEX1KMT2A
SCHEMBL8554060 0.89 KDM4E (0.63) TDP1KDM4EALOX15APEX1KMT2A
SCHEMBL9582012 0.84 TDP1 (0.80) TDP1KDM4EALOX15APEX1KMT2A
SCHEMBL8553783 0.83 HTR1A (0.81) HTR1ADRD2
SCHEMBL8871477 0.82 HTR1A (0.63) TDP1KDM4EALOX15APEX1KMT2A
SCHEMBL8555542 0.82 TDP1 (0.71) TDP1KDM4EALOX15APEX1KMT2A
SCHEMBL8558887 0.81 HTR1A (0.73) TDP1HTR1ADRD2CYP1A2CYP3A4
SCHEMBL8555410 0.80 HTR1A (0.52) HTR1ADRD2
SCHEMBL8554084 0.79 HTR1A (0.78) HTR1ADRD2DRD3
SCHEMBL9581509 0.78 TDP1 (0.79) TDP1KDM4EALOX15APEX1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683166-B1 3-Indolylpiperidines MERCK PATENT GMBH (DE) 1998-10-28 EP disclosed
EP-0683166-A1 3-Indolylpiperidines MERCK PATENT GmbH (DE) 1995-11-22 EP disclosed