SCHEMBL8553222

SCHEMBL8553222

CCC(=O)CC(c1cccnc1)c1ccc2cc(OCOC)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.49
FFAR1 O14842 2/20 0.43
AKR1C3 P42330 4/20 0.41
AKR1C2 P52895 4/20 0.41
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
CYP3A4 P08684 7/20 0.39
CYP26A1 O43174 5/20 0.39
AKR1C1 Q04828 1/20 0.39
PTGS1 P23219 1/20 0.39
CYP2D6 P10635 2/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551198 0.84 CYP3A4 (0.52) PDE4DCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL8550178 0.83 PDE4D (0.42) PDE4DAKR1C3AKR1C2CYP19A1CYP11B1
SCHEMBL8555025 0.82 PDE4D (0.52) PDE4DFFAR1CYP19A1CYP11B1CYP11B2
SCHEMBL8313802 0.81 FFAR1 (0.53) PDE4DFFAR1
SCHEMBL8319920 0.79 PDE4D (0.48) PDE4DFFAR1RAB9A
SCHEMBL27539172 0.78 SLC6A2 (0.52) PDE4DCYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8553432 0.72 CYP17A1 (0.55) PDE4DFFAR1CYP19A1
SCHEMBL8317319 0.72 KCNA5 (0.40) PDE4DFFAR1CYP19A1CYP3A4CYP2D6
SCHEMBL8318114 0.71 SMN1; SMN2 (0.57) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9312935 0.71 PDE4D (0.40) PDE4DFFAR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed