SCHEMBL8550178

SCHEMBL8550178

CCC(O)CC(c1cccnc1)c1ccc2cc(OCOC)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.42
CYP11B1 P15538 4/20 0.40
CYP11B2 P19099 4/20 0.40
CYP19A1 P11511 2/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2D6 P10635 2/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
KCNH2 Q12809 2/20 0.40
CYP51A1 Q16850 2/20 0.37
KCNA5 P22460 1/20 0.36
AKR1C3 P42330 4/20 0.36
AKR1C2 P52895 4/20 0.36
AKR1C1 Q04828 1/20 0.36
PTGS1 P23219 1/20 0.36
CYP2C9 P11712 2/20 0.36
CYP17A1 P05093 2/20 0.36
CYP2C19 P33261 1/20 0.36
CYP26A1 O43174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551012 0.89 PDE4D (0.47) PDE4DCYP11B1CYP11B2CYP19A1CYP3A4
SCHEMBL8553222 0.83 PDE4D (0.49) PDE4DCYP11B1CYP11B2CYP19A1CYP3A4
Hydrochloric Acid SCHEMBL8555644 0.81 CYP3A4 (0.44) PDE4DCYP11B1CYP11B2CYP19A1CYP3A4
SCHEMBL8318114 0.74 SMN1; SMN2 (0.57) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL8551240 0.73 SMN1; SMN2 (0.44) PDE4DSLC6A2SLC6A4SLC6A3KCNA5
SCHEMBL8481502 0.73 CYP11B1 (0.40) CYP11B1CYP11B2CYP19A1CYP51A1CYP2C9
SCHEMBL8317319 0.72 KCNA5 (0.40) PDE4DCYP19A1CYP3A4CYP2D6SLC6A2
SCHEMBL8313802 0.71 FFAR1 (0.53) PDE4DKCNA5
SCHEMBL9311940 0.70 HRH1 (0.42) PDE4DCYP19A1CYP3A4CYP2D6SLC6A2
SCHEMBL8319920 0.70 PDE4D (0.48) PDE4DKCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed