SCHEMBL8555025

SCHEMBL8555025

CCC(=O)CC(c1cccnc1)c1ccc2cc(O)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.52
CYP2C9 P11712 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP19A1 P11511 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
KCNH2 Q12809 2/20 0.42
CYP17A1 P05093 1/20 0.40
ITGB3 P05106 3/20 0.40
ITGAV P06756 3/20 0.40
ITGA2B P08514 1/20 0.40
FFAR1 O14842 1/20 0.39
TBXAS1 P24557 1/20 0.39
CTSA P10619 2/20 0.39
LMNA P02545 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551198 0.90 CYP3A4 (0.52) PDE4DCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL8553432 0.85 CYP17A1 (0.55) PDE4DCYP19A1CYP17A1ITGB3ITGAV
SCHEMBL27539172 0.83 SLC6A2 (0.52) PDE4DCYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL8553222 0.82 PDE4D (0.49) PDE4DCYP19A1CYP11B1CYP11B2CYP3A4
Hydrochloric Acid SCHEMBL8555644 0.80 CYP3A4 (0.44) PDE4DCYP2C9HSD17B10CYP19A1CYP11B1
SCHEMBL8552254 0.74 SUCNR1 (0.50) PDE4DCYP17A1ITGB3ITGAVITGA2B
SCHEMBL9519691 0.73 L3MBTL1 (0.50) PDE4DITGB3ITGAVITGA2BTBXAS1
SCHEMBL3413768 0.68 LMNA (0.55) CYP2D6FFAR1LMNAHPGD
SCHEMBL2303019 0.68 CCNC (0.48) PDE4DCYP3A4TBXAS1CTSALMNA
SCHEMBL17591689 0.68 LMNA (0.54) PDE4DSLC6A2SLC6A4SLC6A3TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed