SCHEMBL8553241

SCHEMBL8553241

CCN(C(=O)CBr)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
PTPN1 P18031 1/20 0.44
TSHR P16473 3/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 1/20 0.43
LTB4R2 Q9NPC1 1/20 0.40
POLB P06746 1/20 0.40
APEX1 P27695 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
HTT P42858 1/20 0.39
MLYCD O95822 3/20 0.39
OPRM1 P35372 1/20 0.39
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21785057 0.85 OPRM1 (0.49) SMN1; SMN2TSHRALDH1A1GLALTB4R2
SCHEMBL8443789 0.84 SMN1; SMN2 (0.47) SMN1; SMN2TSHRALDH1A1GLALTB4R2
SCHEMBL16110560 0.82 MEN1 (0.44) TSHRALDH1A1GLATDP1MLYCD
SCHEMBL8439833 0.82 NPC1 (0.46) SMN1; SMN2TSHRALDH1A1GLALTB4R2
SCHEMBL3138023 0.81 ALDH1A1 (0.66) SMN1; SMN2TSHRALDH1A1GLAMAPT
SCHEMBL5045338 0.79 ALDH1A1 (0.47) SMN1; SMN2TSHRALDH1A1GLAMAPK1
SCHEMBL20964605 0.79 LTB4R2 (0.45) SMN1; SMN2TSHRALDH1A1GLALTB4R2
SCHEMBL5045325 0.78 ALDH1A1 (0.46) SMN1; SMN2TSHRALDH1A1GLALTB4R2
SCHEMBL8552126 0.78 POLQ (0.48) PTPN1KDM4EGAAMAPTKMT2A
Hydrochloric Acid SCHEMBL28795770 0.76 ALDH1A1 (0.44) SMN1; SMN2TSHRALDH1A1GLAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672037-B1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LTD (GB) 1998-07-08 EP disclosed
US-5569654-A ADMINISTERING AS ANTAGONISTS OF GASTRIN AND CHOLECYSTOKININ GLAXO GROUP LIMITED (GB) 1996-10-29 US disclosed
EP-0672037-A1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LIMITED (GB) 1995-09-20 EP disclosed
CN-1093085-A Sulfonamide derivatives GLAXO GROUP LTD (GB) 1994-10-05 CN disclosed
WO-1994013648-A1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LIMITED (GB) 1994-06-23 WO disclosed