SCHEMBL8553701

SCHEMBL8553701

CC(C)(C)CN1CCC(c2csc3ccc(NC(=O)CCCCOc4ccccc4)cc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.43
HTR1D P28221 8/20 0.42
HTR1B P28222 8/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MCHR1 Q99705 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GAA P10253 1/20 0.40
NAMPT P43490 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553620 0.84 DRD2 (0.46) HTR1DHTR1BMAPTALOX15L3MBTL1
SCHEMBL7478444 0.84 HTR1D (0.63) HTR1DHTR1B
SCHEMBL8550557 0.83 DRD2 (0.43) HTR1DHTR1BSMN1; SMN2MAPTMCHR1
SCHEMBL8547605 0.82 RORC (0.45) HTR1DHTR1B
SCHEMBL7484304 0.79 HTR1D (0.58) HTR1DHTR1B
SCHEMBL8548534 0.79 DRD2 (0.48) SMN1; SMN2MAPTALDH1A1CYP1A2CYP3A4
SCHEMBL8547656 0.77 KDM4E (0.45) SMN1; SMN2MAPTL3MBTL1ALDH1A1GAA
SCHEMBL8547532 0.76 BCHE (0.51) BCHEHTR1DHTR1B
SCHEMBL8547952 0.76 HTR1D (0.45) BCHEHTR1DHTR1BSMN1; SMN2ALDH1A1
SCHEMBL8594485 0.76 DRD2 (0.40) HTR1DHTR1BSMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed