SCHEMBL8548534

SCHEMBL8548534

CC(C)(C)CN1CCC(c2coc3ccc(NC(=O)CCOc4ccccc4)cc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.48
HTR2A P28223 16/20 0.48
DRD3 P35462 16/20 0.48
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553620 0.95 DRD2 (0.46) DRD2HTR2ADRD3MAPT
SCHEMBL8548196 0.84 DRD2 (0.52) DRD2HTR2ADRD3
SCHEMBL7484304 0.83 HTR1D (0.58) DRD2
SCHEMBL30909276 0.81 RAB9A (0.42) DRD2HTR2ADRD3RAB9ANPC1
SCHEMBL8387125 0.81 RAB9A (0.42) DRD2HTR2ADRD3RAB9ANPC1
SCHEMBL8708281 0.81 DRD2 (0.45) DRD2HTR2ADRD3
SCHEMBL8553701 0.79 BCHE (0.43) ALDH1A1CYP1A2CYP3A4CYP2D6MAPT
SCHEMBL7478444 0.79 HTR1D (0.63) DRD2
SCHEMBL8594882 0.77 DRD2 (0.45) DRD2HTR2ADRD3
SCHEMBL8551233 0.73 DRD2 (0.46) DRD2HTR2ADRD3KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed