SCHEMBL8553755

SCHEMBL8553755

Cc1ccnc(N2CCN(C(=O)Cc3cn4c5c(cccc35)CCC4)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
MTNR1A P48039 5/20 0.46
MTNR1B P49286 5/20 0.46
KDM4E B2RXH2 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
MAPT P10636 1/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
ALDH1A1 P00352 3/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KMT2A Q03164 1/20 0.42
ALOX5 P09917 1/20 0.42
CPT2 P23786 1/20 0.41
CPT1A P50416 1/20 0.41
CPT1B Q92523 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556855 0.82 ALOX5 (0.54) MTNR1AMTNR1BHTR2AHTR2CALOX5
Hydrochloric Acid SCHEMBL8597178 0.81 ALOX5 (0.53) MTNR1AMTNR1BHTR2AHTR2CALOX5
SCHEMBL8554233 0.79 ALOX5 (0.53) PARP1KDM4ESMN1; SMN2LMNAHTT
SCHEMBL9304984 0.77 ALOX5 (0.45) PARP1KDM4ESMN1; SMN2LMNAHTT
SCHEMBL8552282 0.77 ALOX5 (0.59) PARP1KDM4ESMN1; SMN2LMNAHTT
SCHEMBL8553891 0.73 ALOX5 (0.46) PARP1KDM4ESMN1; SMN2LMNAHTT
SCHEMBL8554489 0.73 PARP1 (0.42) PARP1KDM4ESMN1; SMN2LMNAHTT
SCHEMBL9303578 0.72 HTR2A (0.63) MTNR1AMTNR1BHTR2AHTR2CALDH1A1
SCHEMBL8556392 0.71 ALOX5 (0.59) PARP1KDM4ESMN1; SMN2LMNAHTT
SCHEMBL2260014 0.71 HTR2A (0.65) MTNR1AMTNR1BHTR2AHTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529452-B1 1,7-Condensed 3-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them SOLVAY PHARM GMBH (DE) 1998-11-11 EP disclosed
US-5324725-A Antiinflammatory agent, antiallergen KALI-CHEMIE PHARMA GMBH (DE) 1994-06-28 US disclosed
EP-0529452-A2 1,7-Condensed 2-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them Kali-Chemie Pharma GmbH (DE) 1993-03-03 EP disclosed