SCHEMBL8554030

SCHEMBL8554030

N=C(N)Nc1nnc(-c2ccccc2-c2ccccc2)c2cccc(Br)c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
PLAU P00749 1/20 0.33
PLAT P00750 1/20 0.33
KDR P35968 3/20 0.32
KDM4E B2RXH2 2/20 0.32
THRB P10828 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PLG P00747 1/20 0.32
F9 P00740 1/20 0.32
ENPP3 O14638 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
GRM2 Q14416 1/20 0.31
PDE5A O76074 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8374822 0.90 NPSR1 (0.39) ALDH1A1KDRKDM4ETHRBNPSR1
Hydrochloric Acid SCHEMBL8547376 0.89 NPSR1 (0.39) ALDH1A1KDRKDM4ETHRBNPSR1
SCHEMBL8549269 0.86 HSD11B1 (0.34) KDRMAPTSMN1; SMN2HSD17B10
SCHEMBL8372791 0.86 KDR (0.35) ALDH1A1MAPK1KDRPLGCYP1A2
Hydrochloric Acid SCHEMBL8551586 0.85 KDR (0.34) KDRPLGMAPT
SCHEMBL8552267 0.84 HSD11B1 (0.38) KDRKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8549372 0.83 NPSR1 (0.39) SIGMAR1ALDH1A1PLAUPLATKDR
SCHEMBL8553998 0.80 KDR (0.37) ALDH1A1KDRKDM4ETHRBENPP3
SCHEMBL8549550 0.80 KDR (0.44) ALDH1A1KDRKDM4ENPSR1ENPP3
SCHEMBL8371540 0.78 CCNE2 (0.32) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed