SCHEMBL8552267

SCHEMBL8552267

N=C(N)Nc1nnc(-c2ccccc2C(F)(F)F)c2cccc(Br)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.38
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
RECQL P46063 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
PTPN1 P18031 5/20 0.34
CRHR1 P34998 1/20 0.34
KDR P35968 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EPHX2 P34913 1/20 0.33
DPP4 P27487 1/20 0.32
USP1 O94782 1/20 0.32
WDR48 Q8TAF3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554030 0.84 SIGMAR1 (0.34) CYP1A2CYP2D6CYP2C19CYP3A4HSD17B10
SCHEMBL8549269 0.84 HSD11B1 (0.34) HSD11B1MEN1KMT2AHSD17B10PTPN1
SCHEMBL8372791 0.84 KDR (0.35) CYP1A2CYP2D6CYP2C19KMT2ACYP3A4
Hydrochloric Acid SCHEMBL8551586 0.83 KDR (0.34) KMT2AKDR
SCHEMBL8374822 0.81 NPSR1 (0.39) CYP1A2CYP2D6CYP2C19CYP3A4HSD17B10
SCHEMBL8550319 0.80 KDM4E (0.37) CYP1A2CYP2D6CYP2C19MEN1KMT2A
Hydrochloric Acid SCHEMBL8547376 0.80 NPSR1 (0.39) CYP1A2CYP2D6CYP2C19CYP3A4HSD17B10
Hydrochloric Acid SCHEMBL8548628 0.79 KDM4E (0.37) CYP1A2CYP2D6CYP2C19MEN1KMT2A
SCHEMBL8552274 0.78 PLAU (0.40) HSD11B1
SCHEMBL8553998 0.78 KDR (0.37) CYP1A2CYP2C19MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed