SCHEMBL8554188

SCHEMBL8554188

O=C(O)CCN1CCC(C(=O)Nc2cn(C3CCNCC3)cn2)CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 6/20 0.43
CDK5R1 Q15078 6/20 0.43
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
GSK3B P49841 9/20 0.38
DYRK1A Q13627 8/20 0.38
CPB1 P15086 1/20 0.37
KDM2B Q8NHM5 1/20 0.37
WNT1 P04628 7/20 0.37
S1PR1 P21453 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8618549 0.88 SMN1; SMN2 (0.45) CDK5CDK5R1CARM1PRMT6GSK3B
SCHEMBL8622807 0.78 CARM1 (0.37) CARM1PRMT6GSK3BDYRK1AWNT1
SCHEMBL8554405 0.76 CDK5 (0.47) CDK5CDK5R1GSK3BCPB1KDM2B
Hydrochloric Acid SCHEMBL8551563 0.75 CDK5 (0.38) CDK5CDK5R1GSK3BDYRK1ACPB1
Hydrochloric Acid SCHEMBL8550451 0.72 L3MBTL1 (0.47) CPB1KDM2BITGB3ITGA2B
SCHEMBL8551904 0.71 ALDH1A1 (0.51)
SCHEMBL8141352 0.70 ME3 (0.52) CARM1PRMT6ITGB3ITGA2B
Hydrochloric Acid SCHEMBL8592153 0.69 CDK5 (0.46) CDK5CDK5R1GSK3BDYRK1ACPB1
SCHEMBL1269214 0.68 CDK5 (0.57) CDK5CDK5R1GSK3BKDM2B
Hydrochloric Acid SCHEMBL8621116 0.67 L3MBTL1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed