SCHEMBL8554405

SCHEMBL8554405

O=C(O)CN1CCC(CC(=O)Nc2cn(C3CCNCC3)cn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 9/20 0.47
CDK5R1 Q15078 9/20 0.47
GSK3B P49841 1/20 0.40
DEGS1 O15121 3/20 0.37
USP30 Q70CQ3 2/20 0.37
CPB1 P15086 1/20 0.37
KDM2B Q8NHM5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8592153 0.88 CDK5 (0.46) CDK5CDK5R1GSK3BDEGS1USP30
SCHEMBL8554188 0.76 CDK5 (0.43) CDK5CDK5R1GSK3BCPB1KDM2B
SCHEMBL8551437 0.69 CPB1 (0.37) CPB1KDM2B
SCHEMBL8550443 0.69 CPB1 (0.37) CPB1KDM2B
SCHEMBL8550448 0.69 CPB1 (0.37) CPB1KDM2B
Hydrochloric Acid SCHEMBL8618549 0.69 SMN1; SMN2 (0.45) CDK5CDK5R1GSK3B
SCHEMBL1269214 0.67 CDK5 (0.57) CDK5CDK5R1GSK3BKDM2B
Hydrochloric Acid SCHEMBL8551563 0.67 CDK5 (0.38) CDK5CDK5R1GSK3BCPB1KDM2B
SCHEMBL13406413 0.65 KDM2B (0.49) CDK5CDK5R1CPB1KDM2B
SCHEMBL3282448 0.63 SIGMAR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed